Madame Charline KIEFFER / PhD
Contact details
Professional experience
Jobs
Availability : 1 2015
Mobility : Europe
Research : OUI
PhD
Title : Sciences Chimiques
First registration date : 26 September 2011 / 3A
Doctoral school : Sciences Chimiques - Marseille
Thesis defense date : 11 December 2014
Subject : Pharmacochimie antiprozoaire en séries quinazoline et quinoléine : synthèse, évaluation biologique et recherche de mécanismes d'action
Thesis supervisor : RATHELOT Pascal
Thesis co-supervisor : VERHAEGHE Pierre
Research unit : ICR - Institut de Chimie Radicalaire
Master's degree
Title : Master 2R Chimie
June 2011 - Faculté Saint Jérôme
Mention : Bien
Publications
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Sonogashira cross-coupling reaction in 4-chloro-2-trichloromethylquinazoline series is possible despite a side dimerization reaction
tetrahedron, 2013
Charline Kieffer, Pierre Verhaeghe, Nicolas primas, Caroline Casteras-Ducros, Armand Gellis, Roselyne Rosas, Sylvain Rault, Pascal Rathelot, Patrice Vanelle
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A new synthetic route to original sulfonamide derivatives in 2-trichloromethylquinazoline series: A structure-activity relationship study of antiplasmodial activity.
Molecules, 2012
Nicolas Primas, Pierre Verhaeghe, Anita Cohen, Charline Kieffer, Aurélien Dumètre, Sébastien Hutter, Sylvain Rault, Pascal Rathelot, Nadine Azas, Patrice Vanelle
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Synthesis and biological evaluation of novel trichloromethylpyrrolo[1,2-a]quinoxalines as antiplasmodial agents
European Journal of Medicinal Chemistry, 2014
Nicolas Primas, Peggy Suzanne, Pierre Verhaeghe, Sébastien Hutter, Charline Kieffer, Michèle Laget, Anita Cohen, Julie Broggi, Jean-Charles Lancelot, Aurélien Lesnard, Patrick Dallemagne, Pascal Rathelot, Sylvain Rault, Patrice Vanelle, Nadine Azas.
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Preventing the contamination of hospital personnel by cytotoxic agents: evaluation and training of the PHCWs working in oncology units.
European Journal of Cancer Care, 2014
Charline Kieffer, Pierre Verhaeghe, Sylvie Lagrassa, Régine Grégoire, Zoulikha Moussaoui, Caroline Castera-Ducros, John Elbert Clark, Patrice Vanelle, Pascal Rathelot
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A new DMAP-catalyzed and microwave-assisted approach for introducing 4-heteroarylamino substituents at position 4 of the quinazoline ring
Tetrahedron, 2014
Armand Gellis, Charline Kieffer, Nicolas Primas, Gilles Lanzada, Michel Giorgi, Pierre Verhaeghe, Patrice Vanelle
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Antileishmanial pharmacomodulation in 8-nitroquinolin-2(1H)-one series
Chemmedchem, 2014
Charline Kieffer, Anita Cohen, Pierre Verhaeghe, Lucie Paloque, Sébastien Hutter, Caroline Castera-Ducros, Michèle Laget, Sylvain Rault, Alexis Valentin, Pascal Rathelot,Nadine Azas, Patrice Vanelle
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Looking for new antileishmanial derivatives in 8-nitroquinolin-2(1H)-one series
european journal of medicinal chemistry, 2014
Charline Kieffer,Anita Cohen, Pierre Verhaeghe, Sébastien Hutter, Caroline Castera-Ducros, Michèle Laget, Vincent Remusat, Sylvain Rault, Pascal Rathelot, Nadine Azas, Patrice Vanelle
Languages
Anglais : C1 - Avancé